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Toplam kayıt 7, listelenen: 1-7
Determination of anticancer and antibacterial activities of disubstituted tacrine derivatives
(2019)
The present study describes the biological features of disubstituted tacrine derivatives using cell proliferation andcell cytotoxicity assays. The abilities of tacrine derivatives to inhibit microbial growth and to interact ...
SAR Evaluation of Disubstituted Tacrine Analogues as Promising Cholinesterase and Carbonic Anhydrase Inhibitors
(Assoc Pharmaceutical Teachers India, 2019)
Background: The inhibition of both hydrolysis products of acetylcholine (ACh), Acetylcholinesterase (AChE) and Butyrylcholinesterase (BChE), is essential for successful treatment of Alzhemier patients. Objectives: This ...
Synthesis, characterization, crystal structures, theoretical calculations and biological evaluations of novel substituted tacrine derivatives as cholinesterase and carbonic anhydrase enzymes inhibitors
(Elsevier Science Bv, 2019)
The six and seven hydrocycle membered disilylanilino acridine (tacrine) analogues (9-11) were synthesized by one-pot procedures. The structures of novel silyl tacrine derivatives were characterized by NMR spectroscopy, ...
The adaptation of the pedagogical knowledge and skills survey into Turkish: Validity and reliability study
(Mehmet Tekerek, 2019)
This research aims to adapt the Pedagogical Knowledge and Skills in Teaching (PKST) survey developed by Wong, Chong, Choy and Lim (2012) to Turkish. The participants of the study are 830 4th year students of education ...
Aminopyrazole-substituted metallophthalocyanines: Preparation, aggregation behavior, and investigation of metabolic enzymes inhibition properties
(Wiley-V C H Verlag Gmbh, 2019)
The synthesis, characterization, aggregation behavior, theoretical studies, and investigation of antimicrobial, antidiabetic, and anticholinergic properties of 4-(2-(5-amino-4-(4-bromophenyl)-3-methyl-1H-pyrazol-1-yl)eth ...
4’-Metil-3-Fenilakrilofenon Bileşiğinin Moleküler ve Kristal Yapı Analizi
(2019)
Bileşiğin kristal yapısı (C16H14O) 296 K’de tayin edildi. Tek kristal bileşiğin yapısı tek kristal X-ışını kırınımı yöntemi kullanılarak belirlendi. Kristal yapının birim hücre parametreleri a=14.9921(9) Å, b=9.8460(4) Å, ...
Fen Bilimleri Öğretmenlerinin Teknolojik Pedagojik Alan Bilgilerinin İncelenmesi
(2019)
Bu çalışmanın amacı, fen bilimleri öğretmenlerinin alan bilgilerinin teknoloji ile entegrasyonu sonucunda özyeterlik inançlarını incelemektir. Yapılan çalışmada hem nitel hem de nicel araştırma yöntemlerinden yararlanılmıştır. ...