Konu "SAR" için listeleme
Toplam kayıt 4, listelenen: 1-4
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Farklı implant ve abutment dizaynlarının farklı kemik modelleri üzerinde dikey ve açılı kuvvetler altında meydana getirdiği stres bölgelerinin sonlu elemanlar analizi ile incelenmesi
(Kırıkkale Üniversitesi, 2014)Mekanostatik teorisine göre kemiğe gelen yükleri az olması alveolar kemikte atrofiye neden olurken, yüklerin miktarının fazla olması ise rezorpsiyona neden olabilmektedir. Bu durumdan özellikle normal dişin etrafındaki ... -
SAR Evaluation of Disubstituted Tacrine Analogues as Promising Cholinesterase and Carbonic Anhydrase Inhibitors
(Assoc Pharmaceutical Teachers India, 2019)Background: The inhibition of both hydrolysis products of acetylcholine (ACh), Acetylcholinesterase (AChE) and Butyrylcholinesterase (BChE), is essential for successful treatment of Alzhemier patients. Objectives: This ... -
A SAR Study: Evaluation of Bromo Derivatives of 8-Substituted Quinolines as Novel Anticancer Agents
(Bentham Science Publ Ltd, 2017)Background: Brominated 8-hydroxy, 8-methoxy, 8-amino quinolines 5, 6, 8, 9 and novel cyano 8-hydroxyquinolines 11, 12 were evaluated in vitro for their anticancer effects on various cell lines. 5,7-Dibromo-5, 7-bromo-6, ... -
Synthesis, characterization, and SAR of arylated indenoquinoline-based cholinesterase and carbonic anhydrase inhibitors
(Wiley-V C H Verlag Gmbh, 2018)We report the synthesis of bromoindenoquinolines (15a-f) by Friedlander reactions in low yields (13-50%) and the conversion of the corresponding phenyl-substituted indenoquinoline derivatives 16-21 in high yields (80-96%) ...